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Table 2 BRETMax and BRET50 values from the BRET β-arrestin saturation assay

From: LPA1-mediated inhibition of CXCR4 attenuates CXCL12-induced signaling and cell migration

 

CXCR4-Rluc8 + pcDNA3

CXCR4-Rluc8 + Flag-LPA1

Vehicle

CXCL12

Vehicle

CXCL12

mCitrine- β-arrestin1

ΔBRETMax

0.111

0.198

0.131

0.217

BRET50

8.639

5.273

8.071

8.469

mCitrine- β-arrestin2

ΔBRETMax

0.169

0.383

0.250

0.468

BRET50

4.927

1.564

3.997

2.445