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Table 2 p42/p44 MAP kinase inactivating agents in Prostatic cells

From: Mitogen Activated Protein kinase signal transduction pathways in the prostate

Endogenous

   

Calcitonin

DU145

?

100

15-(S)-HETE

PC3

?

38

Exogenous

   

Lovastatin (HMG-CoA reductase inhibitor)

PC3

?

33

Grape seed extracta

DU145

?

101,102

Methyl selenium molecules

DU145

?

27,103,104

Silibinin

LNCaP, DU145

?

105

Silymarin

DU145

?

51

Genistein

DU145, AT6.3

?

51,106

Kaempferol

AT6.3

?

106

Biochanin A

AT6.3

?

106

Quercetin

PC3

?

91

Phenylacetate

LNCaP

?

34

  1. a Can activate ERK at higher doses