From: Targeting the PDGF signaling pathway in tumor treatment
Inhibitor | Primary targets | Secondary targets |
---|---|---|
Imatinib | Abl, PDGFR, Kit | Raf |
Sunitinib | PDGFR, VEGFR, Kit, Flt3 | Â |
Sorafenib | Raf, VEGFR, PDGFR, Kit, Flt3 | FGFR |
Pazopanib | VEGFR, PDGFR, Kit | FGFR |
Nilotinib | Kit, Abl, PDGFR | Â |
Cediranib | VEGFR, Kit, PDGFR | FGFR |
Motesanib | VEGFR, Kit | PDGFR, Ret |
Axitinib | VEGFR | PDGFR, Kit |
Linifenib | VEGFR, Kit | PDGFR |
Dasatinib | Abl, Src | PDGFR, Kit |
Quizartinib | FLT3 | Kit, PDGFR, Ret, CSF1R |
Ponatinib | Ret, Abl | PDGFR, VEGFR |